SCHEMBL30944945

SCHEMBL30944945

C=CC(=O)Nc1cc(Nc2cc(C(F)(F)F)c3cc(OC)ccc3n2)ccc1OC

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.49
BTK Q06187 2/20 0.47
MAPK3 P27361 4/20 0.45
ERBB3 P21860 2/20 0.42
DUS2 Q9NX74 1/20 0.42
MAPT P10636 1/20 0.42
ERBB2 P04626 1/20 0.42
ERBB4 Q15303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29230158 1.00 EGFR (0.49) EGFRBTKMAPK3ERBB3DUS2
SCHEMBL29230203 0.89 MAPT (0.46) MAPT
SCHEMBL30944970 0.89 MAPT (0.46) MAPT
SCHEMBL29230117 0.83 EGFR (0.46) EGFRMAPT
SCHEMBL30944967 0.83 EGFR (0.46) EGFRMAPT
SCHEMBL30944997 0.83 MEN1 (0.47) MAPT
SCHEMBL29230166 0.83 MEN1 (0.47) MAPT
SCHEMBL30944968 0.81 ABCB1 (0.47) MAPT
SCHEMBL29230132 0.81 ABCB1 (0.47) MAPT
SCHEMBL30945007 0.79 SLC2A1 (0.54) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118146151-A 4-Trifluoromethyl substituted quinoline and quinazoline compound and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2024-06-07 CN disclosed