SCHEMBL30945007

SCHEMBL30945007

COc1ccc2nc(Nc3ccc(NC(C)=O)cc3)cc(C(F)(F)F)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.54
EPHX2 P34913 1/20 0.49
MAPT P10636 9/20 0.48
LMNA P02545 4/20 0.48
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ATM Q13315 1/20 0.47
MTNR1A P48039 3/20 0.47
MTNR1B P49286 3/20 0.47
TP53 P04637 1/20 0.47
BRAF P15056 2/20 0.46
POLB P06746 1/20 0.46
RAD52 P43351 1/20 0.46
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29230224 1.00 SLC2A1 (0.54) SLC2A1EPHX2MAPTLMNAKDM4E
SCHEMBL29230157 0.89 POLB (0.56) SLC2A1MAPTLMNAKDM4EMEN1
SCHEMBL30944961 0.89 POLB (0.56) SLC2A1MAPTLMNAKDM4EMEN1
SCHEMBL30945031 0.89 MAPT (0.52) SLC2A1EPHX2MAPTLMNAKDM4E
SCHEMBL29230179 0.89 MAPT (0.52) SLC2A1EPHX2MAPTLMNAKDM4E
SCHEMBL30944997 0.88 MEN1 (0.47) SLC2A1EPHX2MAPTLMNAKDM4E
SCHEMBL30944970 0.88 MAPT (0.46) SLC2A1MAPTLMNAKDM4EMEN1
SCHEMBL29230203 0.88 MAPT (0.46) SLC2A1MAPTLMNAKDM4EMEN1
SCHEMBL29230166 0.88 MEN1 (0.47) SLC2A1EPHX2MAPTLMNAKDM4E
SCHEMBL30945017 0.86 MAPT (0.54) SLC2A1MAPTLMNAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118146151-A 4-Trifluoromethyl substituted quinoline and quinazoline compound and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2024-06-07 CN disclosed