SCHEMBL30944992

SCHEMBL30944992

COc1ccc2nc(Nc3ccc(C(F)(F)F)cc3)cc(C(F)(F)F)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.52
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
LMNA P02545 3/20 0.52
KDM4E B2RXH2 2/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ACP1 P24666 1/20 0.52
POLB P06746 2/20 0.50
RAD52 P43351 1/20 0.50
GALR2 O43603 1/20 0.49
PKM P14618 1/20 0.47
SLC2A1 P11166 1/20 0.46
PDGFRB P09619 2/20 0.46
PDGFRA P16234 2/20 0.46
GAK O14976 2/20 0.45
KCNH2 Q12809 1/20 0.44
SCN5A Q14524 1/20 0.44
SCN9A Q15858 1/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29230169 1.00 MAPT (0.52) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL29230157 0.94 POLB (0.56) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL30944961 0.94 POLB (0.56) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL30945026 0.90 MEN1 (0.59) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL29230128 0.90 MEN1 (0.59) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL29230131 0.89 MAPT (0.54) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL30945017 0.89 MAPT (0.54) MAPTMEN1KMT2ALMNAKDM4E
Hydrochloric Acid SCHEMBL30945011 0.88 MEN1 (0.48) MAPTMEN1KMT2ALMNAKDM4E
Hydrochloric Acid SCHEMBL29230274 0.88 MEN1 (0.48) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL30944968 0.86 ABCB1 (0.47) MAPTMEN1KMT2ALMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118146151-A 4-Trifluoromethyl substituted quinoline and quinazoline compound and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2024-06-07 CN disclosed