SCHEMBL30945865

SCHEMBL30945865

COc1cccc(CN2CCNC(=O)C2)c1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.58
ALDH1A1 P00352 5/20 0.56
KDM4E B2RXH2 4/20 0.56
KMT2A Q03164 4/20 0.55
CMA1 P23946 1/20 0.54
GAA P10253 1/20 0.53
CHRM3 P20309 1/20 0.49
MEN1 O00255 3/20 0.49
CLPP Q16740 1/20 0.48
OPRM1 P35372 1/20 0.48
ALDH3A1 P30838 1/20 0.48
MAPT P10636 1/20 0.48
ATM Q13315 1/20 0.48
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29234312 1.00 SIGMAR1 (0.58) SIGMAR1ALDH1A1KDM4EKMT2ACMA1
SCHEMBL29194556 0.89 SIGMAR1 (0.47) SIGMAR1ALDH1A1KDM4EKMT2ACMA1
SCHEMBL30245568 0.89 SIGMAR1 (0.47) SIGMAR1ALDH1A1KDM4EKMT2ACMA1
SCHEMBL30245633 0.87 SIGMAR1 (0.47) SIGMAR1ALDH1A1KDM4EKMT2ACMA1
SCHEMBL29194528 0.87 SIGMAR1 (0.47) SIGMAR1ALDH1A1KDM4EKMT2ACMA1
SCHEMBL30245484 0.85 SIGMAR1 (0.44) SIGMAR1ALDH1A1KDM4EKMT2ACMA1
SCHEMBL9871627 0.83 SIGMAR1 (0.60) SIGMAR1ALDH1A1KDM4EKMT2ACMA1
SCHEMBL25205014 0.83 HSD17B10 (0.53) SIGMAR1ALDH1A1KMT2ACMA1GAA
SCHEMBL3847058 0.83 SIGMAR1 (0.72) SIGMAR1ALDH1A1KDM4EKMT2AGAA
SCHEMBL29463795 0.83 SIGMAR1 (0.72) SIGMAR1ALDH1A1KDM4EKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117980302-A Piperazine-based agonists of LFA-1 and VLA-4 德克萨斯心脏研究所 2024-05-03 CN disclosed