SCHEMBL30954505

SCHEMBL30954505

CCOC(=O)c1cc2ncccc2n1CC(C)NC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
GAA P10253 1/20 0.38
HTT P42858 3/20 0.37
HSD17B10 Q99714 2/20 0.37
ABCB1 P08183 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
STING1 Q86WV6 1/20 0.36
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36
CNR2 P34972 1/20 0.35
AAK1 Q2M2I8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27311466 1.00 KDM4E (0.38) KDM4EALDH1A1HPGDGAAHTT
SCHEMBL30954510 0.84 ABCB1 (0.38) KDM4EALDH1A1HPGDGAAHTT
SCHEMBL27311600 0.84 ABCB1 (0.38) KDM4EALDH1A1HPGDGAAHTT
SCHEMBL30954492 0.81 SYK (0.35) KDM4EALDH1A1MEN1KMT2ANPC1
Hydrochloric Acid SCHEMBL30954491 0.80 KDM4E (0.42) KDM4EALDH1A1HPGDHTTHSD17B10
SCHEMBL23092436 0.76 NOD2 (0.41) ALDH1A1GAAMEN1KMT2ANPC1
SCHEMBL29900682 0.76 NOD2 (0.41) ALDH1A1GAAMEN1KMT2ANPC1
SCHEMBL2971266 0.76 SRD5A2 (0.47) MEN1KMT2A
SCHEMBL2984740 0.76 SRD5A2 (0.47) MEN1KMT2A
SCHEMBL2971271 0.76 SRD5A2 (0.47) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024118524-A1 AZAINDOLE COMPOUNDS AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS CEREVEL THERAPEUTICS, LLC (US) 2024-06-06 WO disclosed