SCHEMBL30959535

SCHEMBL30959535

Cc1cc(F)c(C=O)c(Br)c1OC(F)F

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ERN1 O75460 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29344216 0.78 FFAR4 (0.30) ERN1
SCHEMBL21196123 0.77 ERN1 (0.34) ERN1
SCHEMBL29344291 0.76 EPAS1 (0.30)
SCHEMBL30849780 0.74 ERN1 (0.33) ERN1
SCHEMBL31459749 0.74 CYP1A2 (0.36) ERN1
SCHEMBL21216165 0.72 ERN1 (0.39) ERN1
SCHEMBL21195865 0.71 POLB (0.33) ERN1
SCHEMBL29344302 0.71 ERN1 (0.31) ERN1
SCHEMBL16761914 0.71 SRC (0.50) MEN1KMT2A
SCHEMBL25286626 0.70 ERN1 (0.44) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4709371-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2026-03-18 EP disclosed
EP-4615847-A1 SMALL MOLECULE INHIBITORS OF KRAS PROTEINS Merck Sharp & Dohme LLC (US) 2025-09-17 EP disclosed
WO-2024233776-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME LLC (US) 2024-11-14 WO disclosed
WO-2024103010-A1 SMALL MOLECULE INHIBITORS OF KRAS PROTEINS MERCK SHARP & DOHME LLC (US) 2024-05-16 WO disclosed