SCHEMBL30967352

SCHEMBL30967352

CCOC(=O)c1cnc2c(F)cc(SCc3ccccc3)cn12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.45
NPC1 O15118 6/20 0.45
RAB9A P51151 6/20 0.45
ALDH1A1 P00352 5/20 0.45
TSHR P16473 2/20 0.45
NFKB1 P19838 2/20 0.45
NFKB2 Q00653 2/20 0.45
RELA Q04206 2/20 0.45
POLB P06746 3/20 0.40
MAPT P10636 5/20 0.39
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
TDP1 Q9NUW8 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
LMNA P02545 3/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30713240 0.88 SMN1; SMN2 (0.45) SMN1; SMN2NPC1RAB9AALDH1A1TSHR
SCHEMBL29267300 0.88 ALDH1A1 (0.45) SMN1; SMN2NPC1RAB9AALDH1A1TSHR
SCHEMBL30967347 0.86 ALDH1A1 (0.39) SMN1; SMN2NPC1RAB9AALDH1A1POLB
SCHEMBL30967342 0.84 MAPT (0.36) SMN1; SMN2NPC1RAB9AALDH1A1POLB
SCHEMBL31024611 0.82 NPC1 (0.44) SMN1; SMN2NPC1RAB9AALDH1A1TSHR
SCHEMBL31024612 0.82 NPC1 (0.44) SMN1; SMN2NPC1RAB9AALDH1A1TSHR
SCHEMBL30967371 0.76 IDO1 (0.42) SMN1; SMN2NPC1RAB9AALDH1A1PIK3CD
SCHEMBL31258713 0.74 SMN1; SMN2 (0.44) SMN1; SMN2NPC1RAB9AALDH1A1TSHR
SCHEMBL31258785 0.73 ALDH1A1 (0.42) SMN1; SMN2NPC1RAB9AALDH1A1TSHR
SCHEMBL30713218 0.73 NPC1 (0.42) SMN1; SMN2NPC1RAB9AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118459452-B PolyADP ribose hydrolase inhibitor and application thereof 苏州国匡医药科技有限公司 2024-10-25 CN disclosed
WO-2024173514-A1 AMIDE AND ESTER-SUBSTITUTED IMIDAZOPYRIDINE COMPOUNDS IDEAYA BIOSCIENCES, INC. (US) 2024-08-22 WO disclosed
CN-118459452-A PolyADP ribose hydrolase inhibitor and application thereof 苏州国匡医药科技有限公司 2024-08-09 CN disclosed