SCHEMBL30967372

SCHEMBL30967372

CCOC(=O)c1c(SCc2ccccc2)nc2c(F)cccn12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.49
MAPK1 P28482 2/20 0.45
RAB9A P51151 5/20 0.44
MAPT P10636 3/20 0.44
HCRTR1 O43613 1/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.44
ALDH1A1 P00352 8/20 0.43
NPC1 O15118 4/20 0.43
TSHR P16473 2/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30967351 0.83 MAPT (0.39) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL18357777 0.77 SMN1; SMN2 (0.57) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL2866056 0.71 SMN1; SMN2 (0.56) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL2869370 0.71 SMN1; SMN2 (0.55) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL9518825 0.70 MAPK1 (0.70) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL9516836 0.68 MAPK1 (0.67) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL15631933 0.68 SMN1; SMN2 (0.65) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL30902227 0.68 SMN1; SMN2 (0.49) KMT2AMEN1SMN1; SMN2RAB9AMAPT
SCHEMBL2420946 0.68 KDM4E (0.54) SMN1; SMN2KDM4EHSD17B10HTTNPSR1
SCHEMBL7709349 0.67 GAA (0.43) KMT2AMEN1SMN1; SMN2RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118459452-B PolyADP ribose hydrolase inhibitor and application thereof 苏州国匡医药科技有限公司 2024-10-25 CN disclosed
CN-118459452-A PolyADP ribose hydrolase inhibitor and application thereof 苏州国匡医药科技有限公司 2024-08-09 CN disclosed