SCHEMBL30968415

SCHEMBL30968415

COC(=O)[C@H](N)Cc1c(F)c(F)c(C2CNCCN2C(=O)OCc2ccccc2)c(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
HTR2C P28335 1/20 0.41
DPP4 P27487 6/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
DPP7 Q9UHL4 4/20 0.39
PREP P48147 2/20 0.38
PDK1 Q15118 1/20 0.37
PDK2 Q15119 1/20 0.37
PDK3 Q15120 1/20 0.37
PDK4 Q16654 1/20 0.37
CTRB1 P17538 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
ACE2 Q9BYF1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30968466 0.87 PARP1 (0.44) PARP1HTR2CDPP4SMN1; SMN2NPC1
SCHEMBL30968423 0.84 PARP1 (0.48) PARP1HTR2CSMN1; SMN2NPC1RAB9A
SCHEMBL30968480 0.83 PARP1 (0.48) PARP1HTR2CSMN1; SMN2NPC1RAB9A
SCHEMBL30968543 0.79 PARP1 (0.48) PARP1HTR2CSMN1; SMN2NPC1RAB9A
SCHEMBL28567927 0.79 SMN1; SMN2 (0.42) DPP4SMN1; SMN2NPC1RAB9ADPP7
SCHEMBL30968414 0.76 PARP1 (0.40) PARP1HTR2CPREPNPSR1ACE2
SCHEMBL20722816 0.76 SMN1; SMN2 (0.47) HTR2CDPP4SMN1; SMN2NPC1RAB9A
SCHEMBL21685804 0.76 SMN1; SMN2 (0.47) HTR2CDPP4SMN1; SMN2NPC1RAB9A
SCHEMBL2706679 0.75 HTR2C (0.52) PARP1HTR2CSMN1; SMN2NPC1RAB9A
SCHEMBL30968411 0.74 PARP1 (0.45) PARP1HTR2CPREPNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112867712-B Carboxamide as ubiquitin-specific protease inhibitor 瓦洛早期发现股份有限公司 2024-07-16 CN disclosed