SCHEMBL30968414

SCHEMBL30968414

COC1=N[C@H](Cc2c(F)c(F)c(C3CNCCN3C(=O)OCc3ccccc3)c(F)c2F)C(OC)=N[C@H]1C(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
HTR2C P28335 1/20 0.36
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TP53 P04637 1/20 0.34
PREP P48147 1/20 0.34
AADAT Q8N5Z0 1/20 0.34
SIGMAR1 Q99720 7/20 0.33
TMEM97 Q5BJF2 6/20 0.33
ACE2 Q9BYF1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20722634 0.80 SMN1; SMN2 (0.39) HTR2CALDH1A1NPSR1SIGMAR1TMEM97
SCHEMBL30968423 0.78 PARP1 (0.48) PARP1HTR2CNPSR1SIGMAR1TMEM97
SCHEMBL30968480 0.77 PARP1 (0.48) PARP1HTR2CNPSR1PREPSIGMAR1
SCHEMBL30968415 0.76 PARP1 (0.42) PARP1HTR2CNPSR1PREPACE2
SCHEMBL30968466 0.76 PARP1 (0.44) PARP1HTR2CACE2
SCHEMBL30968543 0.73 PARP1 (0.48) PARP1HTR2CNPSR1SIGMAR1TMEM97
SCHEMBL30968411 0.70 PARP1 (0.45) PARP1HTR2CALDH1A1NPSR1PREP
SCHEMBL2706679 0.69 HTR2C (0.52) PARP1HTR2CNPSR1PREPSIGMAR1
SCHEMBL30499783 0.67 PREP (0.42) PARP1HTR2CPREPAADATSIGMAR1
SCHEMBL21129022 0.67 ALDH1A1 (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112867712-B Carboxamide as ubiquitin-specific protease inhibitor 瓦洛早期发现股份有限公司 2024-07-16 CN disclosed