SCHEMBL30985188

SCHEMBL30985188

COC(=O)c1cnc2[nH]ccc2c1Cl

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AXL P30530 6/20 0.55
PRKCI P41743 1/20 0.55
NUDT1 P36639 1/20 0.46
MAP2K1 Q02750 1/20 0.46
TTBK1 Q5TCY1 1/20 0.45
TTBK2 Q6IQ55 1/20 0.45
JAK1 P23458 5/20 0.43
JAK3 P52333 5/20 0.43
CDK8 P49336 1/20 0.42
MGLL Q99685 2/20 0.42
NR4A2 P43354 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2115690 1.00 AXL (0.55) AXLPRKCINUDT1MAP2K1TTBK1
SCHEMBL20956198 0.86 AXL (0.50) AXLPRKCINUDT1JAK1JAK3
SCHEMBL566667 0.86 NUDT1 (0.65) AXLPRKCINUDT1JAK1JAK3
SCHEMBL29477133 0.86 NUDT1 (0.65) AXLPRKCINUDT1JAK1JAK3
SCHEMBL30823440 0.86 AXL (0.50) AXLPRKCINUDT1MAP2K1JAK1
SCHEMBL20956169 0.86 AXL (0.50) AXLPRKCINUDT1MAP2K1JAK1
SCHEMBL31120987 0.85 JAK3 (0.50) AXLPRKCINUDT1JAK1JAK3
SCHEMBL20956013 0.85 JAK3 (0.50) AXLPRKCINUDT1JAK1JAK3
Hydrochloric Acid SCHEMBL29477135 0.85 NUDT1 (0.64) AXLPRKCINUDT1JAK1JAK3
Hydrochloric Acid SCHEMBL29234028 0.85 NUDT1 (0.64) AXLPRKCINUDT1JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118525018-A Bialkyne compound and application thereof 上海艾力斯医药科技股份有限公司 2024-08-20 CN disclosed
WO-2024146502-A1 WEE1 DEGRADING COMPOUNDS BEIJING NEOX BIOTECH LIMITED (CN) 2024-07-11 WO disclosed