SCHEMBL3099207

SCHEMBL3099207

CC(=O)c1ccc(-c2sc(C(N)=O)nc2C)cc1F

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 15/20 0.50
PIK3CD O00329 4/20 0.44
PIK3CA P42336 4/20 0.44
PIK3CG P48736 4/20 0.44
PIK3CB P42338 3/20 0.44
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3075444 0.84 GPR52 (0.47) GPR52PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL2074226 0.80 PIK3CD (0.65) GPR52PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL3099579 0.79 PIK3CG (0.69) PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL2958703 0.78 PIK3CD (0.59) GPR52PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL3164908 0.73 IKBKB (0.38) GPR52PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL688062 0.72 CDC7 (0.46) PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL5048901 0.72 GPR52 (0.56) GPR52
SCHEMBL3156596 0.71 CCNC (0.46) GPR52PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL10367425 0.70 SIRT3 (0.48) PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL3668739 0.70 GPR52 (0.44) GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7799810-B2 Organic compounds NOVARTIS AG (CH) 2010-09-21 US disclosed
US-20100120865-A1 Organic compounds NOVARTIS AG (CH) 2010-05-13 US disclosed
EP-2035413-A2 THIAZOLYL UREA DERIVATIVES AS PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS Novartis AG (CH) 2009-03-18 EP disclosed
WO-2008000421-A2 THIAZOLYL UREA DERIVATIVES AS PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS NOVARTIS AG (CH) 2008-01-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100120865-A1 Organic compounds PIK3C3, PIK3R3, PIK3R4 GPR52 2380/4885PIK3CD 10/4885PIK3CA 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.