SCHEMBL30995018

SCHEMBL30995018

CC(C)(C)OC(=O)c1cn(-c2ccc(Cl)cc2Br)nn1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 8/20 0.45
NOTUM Q6P988 7/20 0.45
KCNMA1 Q12791 1/20 0.42
HDAC8 Q9BY41 1/20 0.41
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRA6 Q16445 1/20 0.38
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15059508 1.00 GPR119 (0.45) GPR119NOTUMKCNMA1HDAC8GABRA1
SCHEMBL16753150 0.86 NOTUM (0.56) NOTUMKCNMA1HDAC8GABRA2
SCHEMBL31234511 0.86 NOTUM (0.56) NOTUMKCNMA1HDAC8GABRA2
SCHEMBL30994998 0.81 NOTUM (0.52) NOTUMKCNMA1HDAC8GABRA2
SCHEMBL16753902 0.81 NOTUM (0.52) NOTUMKCNMA1HDAC8GABRA2
SCHEMBL16754018 0.80 NOTUM (0.53) NOTUMKCNMA1HDAC8
SCHEMBL30995043 0.80 NOTUM (0.53) NOTUMKCNMA1HDAC8
SCHEMBL24624555 0.78 GPR119 (0.40) GPR119NOTUMKCNMA1GABRA1GABRG2
SCHEMBL29772920 0.78 GPR119 (0.40) GPR119NOTUMKCNMA1GABRA1GABRG2
SCHEMBL31123904 0.77 NOTUM (0.41) GPR119NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118894814-A Preparation method of 1- (2-bromo-4-chlorophenyl) -4- (trifluoromethyl) -1H-1,2, 3-triazole 上海康鹏科技股份有限公司 2024-11-05 CN disclosed
CN-118126046-A Substituted macrocyclic compound, and preparation method and application thereof 深圳信立泰药业股份有限公司 2024-06-04 CN disclosed