SCHEMBL31000293

SCHEMBL31000293

CNC(=O)N1CCNc2cccnc21

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.43
AVPR1A P37288 4/20 0.42
GAA P10253 2/20 0.39
PDE2A O00408 4/20 0.39
GPR6 P46095 2/20 0.38
CDK9 P50750 1/20 0.37
TP53 P04637 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7368183 0.78 AVPR1A (0.54) AVPR1A
SCHEMBL30454811 0.77 MAPK1 (0.53) AVPR1A
SCHEMBL12405333 0.72 MEN1 (0.38) AVPR1A
SCHEMBL11587275 0.69 NPSR1 (0.49) GAA
SCHEMBL12723718 0.68 AVPR1A (0.41) AVPR1AGAAPDE2ATP53
SCHEMBL20571416 0.68 JAK2 (0.40) AVPR1A
SCHEMBL3920302 0.68 PARP1 (0.38) CYP11B2KCNH2
SCHEMBL26547297 0.68 EPHX2 (0.39) AVPR1AGAA
SCHEMBL19644152 0.67 MAPK1 (0.61) TP53
SCHEMBL7017304 0.66 MEN1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3630770-B1 PYRAZOLO[3,4-B]PYRAZINE DERIVATIVES AS SHP2 PHOSPHATASE INHIBITORS RELAY THERAPEUTICS INC (US) 2024-08-28 EP disclosed