SCHEMBL30454811

SCHEMBL30454811

CC(C)(C)OC(=O)N1CCNc2cccnc21

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.53
POLB P06746 1/20 0.45
GPR119 Q8TDV5 4/20 0.41
AVPR1A P37288 4/20 0.40
GRM5 P41594 3/20 0.39
GRM1 Q13255 2/20 0.39
DTYMK P23919 1/20 0.39
AKT1 P31749 1/20 0.38
KIT P10721 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29505992 0.80 MAPK1 (0.60) MAPK1GPR119AVPR1A
SCHEMBL975814 0.80 MAPK1 (0.60) MAPK1GPR119AVPR1A
SCHEMBL12473225 0.80 PDE2A (0.52) MAPK1POLB
SCHEMBL30462275 0.78 POLB (0.47) MAPK1POLBGPR119GRM5GRM1
SCHEMBL31000293 0.77 CYP11B2 (0.43) AVPR1A
SCHEMBL31357123 0.76 MAPK1 (0.53) MAPK1POLBGPR119AVPR1A
SCHEMBL861264 0.76 POLB (0.45) MAPK1POLBGPR119GRM5GRM1
SCHEMBL31170824 0.76 MAPK1 (0.53) MAPK1POLBGPR119AVPR1A
SCHEMBL1351555 0.76 MAPK1 (0.47) MAPK1POLBGPR119GRM5GRM1
SCHEMBL1092663 0.75 POLB (0.44) POLBGPR119GRM5GRM1DTYMK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478211-B Novel CGRP receptor antagonist and application thereof 石家庄迪斯凯威医药科技有限公司 2023-10-24 CN disclosed
CN-116478211-A Novel CGRP receptor antagonist and application thereof 石家庄迪斯凯威医药科技有限公司 2023-07-25 CN disclosed