SCHEMBL31017347

SCHEMBL31017347

COCCn1ncc2ccc(NC(=O)OC(C)(C)C)c(OC)c21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
GSK3B P49841 1/20 0.37
DYRK1A Q13627 1/20 0.37
PDE10A Q9Y233 2/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ABL1 P00519 2/20 0.33
SRC P12931 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
ATM Q13315 1/20 0.33
NR1I2 O75469 1/20 0.33
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30895142 1.00 MAPK1 (0.38) MAPK1MAOAMAOBGSK3BDYRK1A
SCHEMBL25750456 0.90 GSK3B (0.37) MAPK1GSK3BDYRK1AKDM4ENPC1
SCHEMBL31017361 0.90 GSK3B (0.37) MAPK1GSK3BDYRK1AKDM4ENPC1
SCHEMBL25672474 0.88 MAPK1 (0.39) MAPK1GSK3BDYRK1AKDM4EABL1
SCHEMBL25758055 0.86 KDM4E (0.36) GSK3BDYRK1AKDM4ENPC1RAB9A
SCHEMBL30895063 0.86 MAPK1 (0.38) MAPK1GSK3BDYRK1AABL1SRC
SCHEMBL27199684 0.85 MAPK1 (0.43) MAPK1MAOAMAOBPDE10AKDM4E
SCHEMBL30860930 0.84 GSK3B (0.40) MAPK1GSK3BDYRK1AABL1HTT
SCHEMBL25756633 0.84 GSK3B (0.40) MAPK1GSK3BDYRK1AABL1HTT
SCHEMBL30895022 0.84 HTR2A (0.36) MAPK1GSK3BDYRK1AABL1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118401516-A TYK2 inhibitors, compositions and methods thereof 凌科药业(杭州)有限公司 2024-07-26 CN disclosed