SCHEMBL31028385

SCHEMBL31028385

NC(=O)n1ccnc1-c1nccs1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.35
PARP1 P09874 1/20 0.35
ALDH1A1 P00352 2/20 0.34
PDPK1 O15530 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
ABL1 P00519 1/20 0.34
BCR P11274 1/20 0.34
GRIK1 P39086 1/20 0.34
GRIA1 P42261 1/20 0.34
GRIA2 P42262 1/20 0.34
GRIA3 P42263 1/20 0.34
GRIA4 P48058 1/20 0.34
GRIK2 Q13002 1/20 0.34
GRIK3 Q13003 1/20 0.34
GRIK4 Q16099 1/20 0.34
GRIK5 Q16478 1/20 0.34
ADORA1 P30542 1/20 0.33
HSP90AA1 P07900 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3065487 0.71 ESR1 (0.40) PDPK1
SCHEMBL446875 0.70
SCHEMBL28193727 0.70 PDPK1 (0.34) ALDH1A1PDPK1LOXL2ADORA1HSP90AA1
SCHEMBL27608927 0.69 PDPK1 (0.39) ALDH1A1PDPK1LOXL2ADORA1HSP90AA1
SCHEMBL12320187 0.69 ADORA2A (0.43) PDPK1LOXL2ADORA1HSP90AA1HPGD
SCHEMBL10668273 0.69 ESR1 (0.51) PARP1ALDH1A1HDAC4
Hydrochloric Acid SCHEMBL16433303 0.69 PARP1 (0.42) PARP1ALDH1A1CYP3A4TSHRNOS1
SCHEMBL3055990 0.67 AGTR2 (0.43) ALDH1A1HSP90AA1ECE1
SCHEMBL28750902 0.67 AGTR2 (0.39) ALDH1A1HSP90AA1ECE1
SCHEMBL12276988 0.67 HPGD (0.38) PDPK1LOXL2ADORA1HSP90AA1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3892272-B1 BIFUNCTIONAL MOLECULES FOR DEGRADATION OF EGFR AND METHODS OF USE DANA FARBER CANCER INST INC (US) 2024-07-24 EP disclosed