SCHEMBL31035573

SCHEMBL31035573

FC(F)(F)c1ccn2cc(C(Cl)Cl)nc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
USP7 Q93009 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.33
NPC1 O15118 3/20 0.33
NFKB1 P19838 3/20 0.33
RAB9A P51151 3/20 0.33
NFKB2 Q00653 3/20 0.33
RELA Q04206 3/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RECQL P46063 1/20 0.33
CA2 P00918 1/20 0.33
MCHR1 Q99705 2/20 0.33
TRPA1 O75762 1/20 0.33
MAPT P10636 1/20 0.31
KDM4E B2RXH2 3/20 0.30
ALDH1A1 P00352 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31035876 0.79 PDE10A (0.39) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL720360 0.78 SMN1; SMN2 (0.50) USP7SMN1; SMN2NPC1NFKB1RAB9A
SCHEMBL15767035 0.76 GRM5 (0.44) PARP1SMN1; SMN2MCHR1
SCHEMBL12777909 0.76 PARP1 (0.38) PARP1USP7SMN1; SMN2NPC1NFKB1
SCHEMBL1905278 0.75 KDM4E (0.38) PARP1USP7SMN1; SMN2NPC1RAB9A
SCHEMBL19497542 0.73 MCHR1 (0.44) PARP1USP7SMN1; SMN2CA2MCHR1
SCHEMBL23530832 0.72 NOTUM (0.43) PARP1USP7SMN1; SMN2NPC1RAB9A
SCHEMBL4889270 0.72 PARP1 (0.39) PARP1USP7SMN1; SMN2NPC1NFKB1
SCHEMBL25670702 0.72 KDM4E (0.41) PARP1USP7SMN1; SMN2NPC1RAB9A
SCHEMBL28535736 0.71 TLR9 (0.57) PARP1SMN1; SMN2NPC1NFKB1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118434744-A Nitrogen-containing macrocyclic compound, and preparation method and medical application thereof 中国医药研究开发中心有限公司 2024-08-02 CN disclosed