SCHEMBL31037441

SCHEMBL31037441

CC(C)(C)OC(=O)N(c1cc(Br)ccc1C#N)C(C(=O)O)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.41
TRPA1 O75762 1/20 0.35
CTSS P25774 3/20 0.34
CTSK P43235 3/20 0.34
CTSB P07858 1/20 0.34
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SLC22A12 Q96S37 1/20 0.31
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28885597 0.77 AAK1 (0.43) AAK1TRPA1CTSSCTSKCTSB
SCHEMBL23727009 0.75 AAK1 (0.43) AAK1TRPA1CTSSCTSKCTSB
SCHEMBL31320985 0.75 CTSB (0.36) AAK1CTSSCTSKCTSBSMN1; SMN2
SCHEMBL23750733 0.73 AAK1 (0.42) AAK1TRPA1CTSSCTSKCTSB
SCHEMBL16794066 0.70 AAK1 (0.45) AAK1TRPA1CTSSCTSKCTSB
SCHEMBL4797996 0.70 PTPN1 (0.36) TRPA1CTSSCTSKCTSBSMN1; SMN2
SCHEMBL4797998 0.70 PTPN1 (0.36) TRPA1CTSSCTSKCTSBSMN1; SMN2
SCHEMBL30808724 0.70 PTPN1 (0.36) TRPA1CTSSCTSKCTSBSMN1; SMN2
Water SCHEMBL29079149 0.68 AAK1 (0.44) AAK1CTSSCTSKCTSB
SCHEMBL16809840 0.68 AAK1 (0.45) AAK1TRPA1CTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115335380-B Tricyclic heteroaryl compounds useful as IRAK4 inhibitors 百时美施贵宝公司 2024-08-02 CN disclosed