SCHEMBL31049778

SCHEMBL31049778

Cc1cccnc1-c1ccc(Br)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.51
CYP2A6 P11509 2/20 0.47
TRPV1 Q8NER1 3/20 0.43
SMO Q99835 1/20 0.40
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
NPC1 O15118 3/20 0.38
MAPK1 P28482 2/20 0.38
RAB9A P51151 2/20 0.38
TP53 P04637 1/20 0.38
CNR2 P34972 1/20 0.37
TGFBR1 P36897 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31049777 1.00 METAP2 (0.51) METAP2CYP2A6TRPV1SMONOS3
SCHEMBL11927612 0.81 CCR1 (0.56) METAP2CYP2A6TRPV1NOS3NOS1
SCHEMBL28453842 0.79 METAP2 (0.51) METAP2CYP2A6TRPV1SMONOS3
SCHEMBL26422208 0.78 CCR1 (0.35) CYP2A6NPC1MAPK1RAB9ATP53
SCHEMBL4383276 0.78 S1PR1 (0.37) NPC1MAPK1RAB9ATP53KDM4E
SCHEMBL10112296 0.76 TRPV1 (0.64) METAP2CYP2A6TRPV1NOS3NOS1
SCHEMBL29531176 0.75 KDM4E (0.60) METAP2CYP2A6NOS3NOS1NOS2
SCHEMBL230048 0.75 KDM4E (0.60) METAP2CYP2A6NOS3NOS1NOS2
SCHEMBL2005454 0.74 IDO1 (0.46) METAP2NPC1MAPK1RAB9ATP53
SCHEMBL17992229 0.73 COMT (0.40) NPC1MAPK1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024166133-A1 LIGAND SCAFFOLD FOR PROXIMAL & REMOTE BORYLATION OF ARENES CENTRE OF BIOMEDICAL RESEARCH (IN) 2024-08-15 WO disclosed