SCHEMBL31064012

SCHEMBL31064012

Cc1cc(NC2CCN(C(=O)OCC3CCCN3C(=O)/C=C/CN(C)C)CC2)n2ncc(C(C)C)c2n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK7 P50613 7/20 0.71
CDK9 P50750 2/20 0.71
CDK4 P11802 1/20 0.71
CCNH P51946 6/20 0.42
MNAT1 P51948 6/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
BTK Q06187 5/20 0.36
EGFR P00533 4/20 0.36
LCK P06239 3/20 0.36
ITK Q08881 3/20 0.36
CDK2 P24941 4/20 0.35
GSK3B P49841 1/20 0.35
JAK3 P52333 1/20 0.34
NPC1 O15118 1/20 0.34
NR2F2 P24468 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31064033 0.89 CDK7 (0.57) CDK7CDK9CDK4CCNHMNAT1
SCHEMBL31064241 0.85 CDK9 (0.54) CDK7CDK9CDK4MEN1KMT2A
SCHEMBL21539654 0.83 CDK7 (1.00) CDK7CDK9CDK4CCNHMNAT1
SCHEMBL20971696 0.83 CDK7 (1.00) CDK7CDK9CDK4CCNHMNAT1
SCHEMBL20971700 0.83 CDK7 (1.00) CDK7CDK9CDK4CCNHMNAT1
SCHEMBL20971695 0.83 CDK7 (1.00) CDK7CDK9CDK4CCNHMNAT1
Hydrochloric Acid SCHEMBL20971692 0.82 CDK7 (0.98) CDK7CDK9CDK4CCNHMNAT1
Water SCHEMBL29788116 0.80 CDK7 (0.89) CDK7CDK9CDK4CCNHMNAT1
SCHEMBL31064124 0.80 CDK7 (0.59) CDK7CDK9CDK4CCNHMNAT1
SCHEMBL20971702 0.78 CDK7 (0.85) CDK7CDK9CDK4CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175024-A1 NEW FUSED HETEROCYCLIC COMPOUND AS CDKS INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2024-08-29 WO disclosed