SCHEMBL31067688

SCHEMBL31067688

COc1cc2ncnc(Nc3ccc(NC(=O)Nc4ccccc4C)cc3)c2cc1OC

nearest known ligand 0.80

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.80
EGFR P00533 9/20 0.74
KIT P10721 1/20 0.69
AURKA O14965 1/20 0.68
AURKB Q96GD4 1/20 0.68
MAPK14 Q16539 1/20 0.67
PDGFRA P16234 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31067670 0.92 KDR (0.84) KDREGFRKITAURKAAURKB
SCHEMBL31067653 0.89 KDR (0.79) KDREGFRKITAURKAAURKB
SCHEMBL31067741 0.89 KDR (0.79) KDREGFRKITAURKAAURKB
SCHEMBL31067668 0.89 KDR (0.79) KDREGFRKITAURKAAURKB
SCHEMBL31067691 0.89 KDR (0.79) KDREGFRKITAURKAAURKB
SCHEMBL31067650 0.87 KDR (0.83) KDREGFRKITAURKAAURKB
SCHEMBL31067640 0.85 KDR (0.84) KDREGFRKITAURKAAURKB
SCHEMBL31067666 0.85 KDR (1.00) KDREGFRKITAURKAAURKB
SCHEMBL6163604 0.85 KDR (0.64) KDREGFRAURKAAURKBMAPK14
SCHEMBL6165277 0.85 KDR (0.64) KDREGFRAURKAAURKBMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118530175-A PDGFR inhibitor and preparation method and application thereof 中国药科大学 2024-08-23 CN disclosed