SCHEMBL31067640

SCHEMBL31067640

COc1cc2ncnc(Nc3ccc(NC(=O)Nc4ccc(Br)cc4)cc3)c2cc1OC

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.84
EGFR P00533 7/20 0.84
KIT P10721 1/20 0.84
AURKA O14965 1/20 0.69
AURKB Q96GD4 1/20 0.69
HDAC3 O15379 1/20 0.69
HDAC4 P56524 1/20 0.69
HDAC1 Q13547 1/20 0.69
HDAC7 Q8WUI4 1/20 0.69
HDAC2 Q92769 1/20 0.69
HDAC10 Q969S8 1/20 0.69
HDAC11 Q96DB2 1/20 0.69
HDAC8 Q9BY41 1/20 0.69
HDAC6 Q9UBN7 1/20 0.69
HDAC9 Q9UKV0 1/20 0.69
HDAC5 Q9UQL6 1/20 0.69
BRAF P15056 1/20 0.68
GAK O14976 1/20 0.68
RIPK2 O43353 1/20 0.68
STK10 O94804 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31067695 0.92 KDR (1.00) KDREGFRKITHDAC3HDAC4
SCHEMBL31067666 0.91 KDR (1.00) KDREGFRKITAURKAAURKB
SCHEMBL31067650 0.91 KDR (0.83) KDREGFRKITAURKAAURKB
SCHEMBL5467825 0.90 EGFR (1.00) KDREGFRGAKRIPK2STK10
SCHEMBL31067708 0.90 KDR (0.82) KDREGFRKITAURKAAURKB
SCHEMBL31067633 0.90 KDR (0.82) KDREGFRKITAURKAAURKB
SCHEMBL31067662 0.90 EGFR (0.82) KDREGFRKITAURKAAURKB
Hydrochloric Acid SCHEMBL5479908 0.89 EGFR (0.97) KDREGFRGAKRIPK2STK10
SCHEMBL31067691 0.88 KDR (0.79) KDREGFRKITAURKAAURKB
SCHEMBL31067608 0.87 KDR (0.85) KDREGFRKITAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118530175-A PDGFR inhibitor and preparation method and application thereof 中国药科大学 2024-08-23 CN disclosed