SCHEMBL31068950

SCHEMBL31068950

C=C(C)c1ccncc1N

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
TDP1 Q9NUW8 2/20 0.57
KDM4C Q9H3R0 2/20 0.57
MAPT P10636 2/20 0.57
MEN1 O00255 1/20 0.57
KDM6B O15054 1/20 0.57
KDM4A O75164 1/20 0.57
THRB P10828 1/20 0.57
KMT2A Q03164 1/20 0.57
KDM4D Q6B0I6 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
GAA P10253 2/20 0.55
GLA P06280 1/20 0.55
AOC1 P19801 2/20 0.41
AOC3 Q16853 2/20 0.41
SIRT3 Q9NTG7 1/20 0.37
EP300 Q09472 1/20 0.37
KAT2B Q92831 1/20 0.37
KAT8 Q9H7Z6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31068868 0.83 GAA (0.43) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL16852630 0.80 TDP1 (0.41) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL13299970 0.79 KDM4C (0.68) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL31139848 0.79 KDM4C (0.68) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL19142257 0.79 KDM4E (0.57) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL526501 0.75 CCNC (0.36) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL5700488 0.75 GAA (0.43) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL5700390 0.75 MAPT (0.39) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL19273667 0.75 LOXL2 (0.39) KDM4EALDH1A1TDP1KDM4CMAPT
SCHEMBL29741235 0.75 TDP1 (0.59) KDM4EALDH1A1TDP1KDM4CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12616682-B2 1-H-pyrrolo[2,3-c]pyridine compounds ACERTA PHARMA B.V. (NL) 2026-05-05 US disclosed
EP-4688776-A1 1-H-PYRROLO[2,3-C]PYRIDINE COMPOUNDS ACTING AGAINST CANCER VIA AGONISM OF MENIN Acerta Pharma B.V. (NL) 2026-02-11 EP disclosed
US-20250360112-A1 1-H-PYRROLO[2,3-c]PYRIDINE COMPOUNDS ACERTA PHARMA BV (NL) 2025-11-27 US disclosed
US-20240335431-A1 1-H-PYRROLO[2,3-c]PYRIDINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2024-10-10 US disclosed
WO-2024201240-A1 1-H-PYRROLO[2,3-C]PYRIDINE COMPOUNDS ACTING AGAINST CANCER VIA AGONISM OF MENIN ACERTA PHARMA B.V. (NL) 2024-10-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12616682-B2 1-H-pyrrolo[2,3-c]pyridine compounds MEN1, PKD1, PKD2 KDM4E 308/4885ALDH1A1 1116/4885TDP1 2754/4885
US-20240335431-A1 1-H-PYRROLO[2,3-c]PYRIDINE COMPOUNDS MEN1, PKD1, ADCYAP1R1 KDM4E 3480/4885ALDH1A1 2614/4885TDP1 1671/4885
US-20250360112-A1 1-H-PYRROLO[2,3-c]PYRIDINE COMPOUNDS MEN1, PKD1, ADCYAP1R1 KDM4E 3480/4885ALDH1A1 2614/4885TDP1 1671/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.