SCHEMBL31069728

SCHEMBL31069728

CNc1nc2cc(-c3cnc4c(c3)C(=O)N(Cc3cc(OC(F)(F)F)ccc3F)CCO4)ccn2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.43
SCN4A P35499 1/20 0.43
KCNH2 Q12809 1/20 0.43
SCN5A Q14524 1/20 0.43
SCN9A Q15858 1/20 0.43
SCN2A Q99250 1/20 0.43
SCN3A Q9NY46 1/20 0.43
SCN8A Q9UQD0 1/20 0.43
SCN10A Q9Y5Y9 1/20 0.43
TNIK Q9UKE5 11/20 0.43
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
ALPL P05186 2/20 0.37
RIPK1 Q13546 5/20 0.35
AURKA O14965 1/20 0.34
FLT1 P17948 1/20 0.34
GCK P35557 1/20 0.34
FLT4 P35916 1/20 0.34
MAP3K11 Q16584 1/20 0.34
STK17A Q9UEE5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25379054 0.92 SCN1A (0.42) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL25379735 0.89 TNIK (0.48) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL31069733 0.89 TNIK (0.48) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL29847299 0.89 TNIK (0.36) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL23753782 0.89 TNIK (0.36) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL25416521 0.79 TNIK (0.54) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL23753851 0.79 RIPK1 (0.36) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL29846792 0.79 RIPK1 (0.36) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL31069717 0.79 TNIK (0.47) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL25380573 0.79 TNIK (0.47) SCN1ASCN4AKCNH2SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118556044-A Fused heterocyclic compound, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2024-08-27 CN disclosed