SCHEMBL31153373

SCHEMBL31153373

CSc1ncc2ccc(=O)n([C@@H]3CCC[C@@H](O)C3)c2n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 15/20 0.58
CCND1 P24385 14/20 0.58
CCNE1 P24864 13/20 0.58
CDK6 Q00534 9/20 0.58
CDK4 P11802 9/20 0.58
CCND3 P30281 6/20 0.58
CCND2 P30279 5/20 0.44
CCNA2 P20248 3/20 0.44
FGFR1 P11362 1/20 0.44
FGFR2 P21802 1/20 0.44
FGFR4 P22455 1/20 0.44
FGFR3 P22607 1/20 0.44
CCNT1 O60563 3/20 0.42
CDK9 P50750 3/20 0.42
CCNA1 P78396 2/20 0.42
MAPK8 P45983 1/20 0.42
MAPK9 P45984 1/20 0.42
MAPK10 P53779 1/20 0.42
JAK2 O60674 2/20 0.41
JAK1 P23458 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19857375 1.00 CDK2 (0.58) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL574660 0.87 CCND1 (0.56) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL29990953 0.87 CCND1 (0.56) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL5263603 0.86 CCND1 (0.57) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL4828470 0.86 CCND1 (0.57) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL31637530 0.84 CCND1 (0.49) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL4828611 0.84 CCND1 (0.49) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL24669667 0.82 CDK2 (0.53) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL19863588 0.81 CCNE1 (0.65) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL29798894 0.81 CCNE1 (0.65) CDK2CCND1CCNE1CDK6CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394966-B Pyridopyrimidinone CDK2/4/6 inhibitors 辉瑞公司 2024-10-11 CN disclosed