SCHEMBL31160271

SCHEMBL31160271

CC(C)(C)OC(=O)Nc1cncc(CO[Si](C)(C)C(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.43
NAMPT P43490 2/20 0.42
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39
MAPK14 Q16539 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA9 Q16790 1/20 0.37
PSMB8 P28062 1/20 0.37
SCD O00767 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
HDAC1 Q13547 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
RORC P51449 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17174926 0.86 KDM4E (0.41) NAMPT
SCHEMBL17161617 0.85 BACE1 (0.33) NAMPTSIRT2
SCHEMBL19022370 0.84 TOP2A (0.41) CYP17A1NAMPTTOP2ATOP2BMAPK14
SCHEMBL2797957 0.84 SIRT2 (0.50) CYP17A1NAMPTTOP2ATOP2BCA12
SCHEMBL31139283 0.84 SIRT2 (0.50) CYP17A1NAMPTTOP2ATOP2BCA12
SCHEMBL12639204 0.83 CYP17A1 (0.55) CYP17A1NAMPTMAPK14CA12CA1
SCHEMBL31160327 0.83 TOP2A (0.43) CYP17A1NAMPTTOP2ATOP2BCA12
SCHEMBL15972019 0.82 CYP17A1 (0.48) CYP17A1NAMPTTOP2ATOP2BMAPK14
SCHEMBL30530906 0.82 CYP17A1 (0.48) CYP17A1NAMPTTOP2ATOP2BMAPK14
SCHEMBL14659184 0.82 RAB9A (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025050636-A1 MACROCYCLIC PYRAZOLOPYRIMIDINE COMPOUND AND USE THEREOF 浙江养生堂天然药物研究所有限公司 2025-03-13 WO disclosed
WO-2024199069-A1 POLYARYL-CONTAINING MACROCYCLIC COMPOUND AND USE THEREOF 浙江养生堂天然药物研究所有限公司 2024-10-03 WO disclosed