SCHEMBL3120101

SCHEMBL3120101

c1ccc(-c2cn(C3CC[N]CC3)nn2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.62
DRD4 P21917 2/20 0.62
DRD3 P35462 1/20 0.62
SRC P12931 2/20 0.52
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
DPP4 P27487 2/20 0.43
XDH P47989 1/20 0.43
CYP19A1 P11511 2/20 0.41
KDM6B O15054 1/20 0.41
KDM4A O75164 1/20 0.41
KDM5C P41229 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM2A Q9Y2K7 1/20 0.41
NAMPT P43490 1/20 0.41
LGALS1 P09382 1/20 0.40
LGALS3 P17931 1/20 0.40
BCHE P06276 1/20 0.40
CHRNB2 P17787 2/20 0.39
CHRNB4 P30926 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301787 0.83 DRD2 (0.60) DRD2DRD4DRD3SRCNPC1
SCHEMBL9551505 0.77 DRD2 (0.54) DRD2DRD4DRD3SRCNPC1
SCHEMBL15441288 0.77 DRD2 (0.54) DRD2DRD4DRD3SRCNPC1
SCHEMBL15441290 0.77 DRD2 (0.54) DRD2DRD4DRD3SRCNPC1
SCHEMBL8482373 0.77 DRD4 (1.00) DRD2DRD4DRD3CYP19A1NAMPT
Hydrochloric Acid SCHEMBL8131385 0.76 DRD2 (0.53) DRD2DRD4DRD3SRCNPC1
SCHEMBL19179891 0.75 DRD2 (0.52) DRD2DRD4DRD3SRCNPC1
SCHEMBL27812294 0.75 DRD2 (0.58) DRD2DRD4DRD3SRCNPC1
SCHEMBL19128795 0.73 DRD2 (0.50) DRD2DRD4DRD3SRCNPC1
SCHEMBL12369621 0.73 DRD2 (0.50) DRD2DRD4DRD3SRCNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010022055-A2 INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS AMGEN INC. (US) 2010-02-25 WO claimed
WO-2010022055-A2 INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS AMGEN INC. (US) 2010-02-25 WO disclosed