Ammonia Solution, Strong

Ammonia Solution, Strong

SCHEMBL3120960

N.Nc1nc(-c2ccccc2)cc(-c2ccc(Cc3ccnc(C(F)(F)F)c3)cc2)n1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.56
HSD17B10 Q99714 2/20 0.56
ADORA2A P29274 3/20 0.48
ADORA1 P30542 1/20 0.48
LOXL2 Q9Y4K0 2/20 0.46
LOX P28300 1/20 0.45
ALDH1A1 P00352 2/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CYP1A1 P04798 1/20 0.44
CYP1B1 Q16678 1/20 0.44
LTA4H P09960 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
AURKA O14965 1/20 0.41
HSP90AA1 P07900 1/20 0.41
PRKACA P17612 1/20 0.41
XDH P47989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1644536 0.86 AGPAT2 (0.54) KDM4EHSD17B10LOXL2LOXHRH4
SCHEMBL1644558 0.76 LOXL2 (0.62) LOXL2LOXALDH1A1CA2CYP3A4
SCHEMBL2991593 0.73 KDM4E (1.00) KDM4EHSD17B10ADORA2AADORA1ALDH1A1
SCHEMBL28013042 0.70 HSP90AA1 (0.71) KDM4EADORA2AADORA1ALDH1A1LTA4H
SCHEMBL19417246 0.69 ADORA2A (0.91) KDM4EHSD17B10ADORA2AADORA1ALDH1A1
SCHEMBL4904514 0.69 ADORA2A (1.00) KDM4EHSD17B10ADORA2AADORA1ALDH1A1
SCHEMBL12728025 0.68 AGPAT2 (0.57) HSD17B10HRH4AURKAMAPK1TP53
SCHEMBL12728030 0.68 AGPAT2 (0.57) HSD17B10ADORA2AADORA1HRH4AURKA
SCHEMBL12728031 0.68 AGPAT2 (0.63) KDM4EHRH4AURKAHSP90AA1TP53
SCHEMBL1644550 0.68 POLB (0.58) KDM4ELOXL2LOXALDH1A1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678804-B2 Pyrimidine derivatives for treatment of hyperproliferative disorders BAYER HEALTHCARE LLC (US) 2010-03-16 US disclosed
US-20050277640-A1 Pyrimidine derivatives for treatment of hyperproliferative disorders BAYER PHARMACEUTICALS CORPORATION (US) 2005-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050277640-A1 Pyrimidine derivatives for treatment of hyperproliferative disorders TYMP, DPYD, CCNA2 KDM4E 2029/4885HSD17B10 3124/4885ADORA2A 809/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.