SCHEMBL31226164

SCHEMBL31226164

Cc1cc(-c2nnc3c(C)c(C)c(Cl)nn23)no1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 10/20 0.43
GABRG2 P18507 10/20 0.43
GABRB3 P28472 10/20 0.43
GABRA5 P31644 10/20 0.43
GABRA3 P34903 10/20 0.43
GABRA2 P47869 10/20 0.43
GABRA4 P48169 2/20 0.43
GABRA6 Q16445 1/20 0.43
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
CACNA2D1 P54289 1/20 0.35
P2RX7 Q99572 2/20 0.35
KDM4E B2RXH2 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1258627 0.81 GABRA1 (0.58) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL31058084 0.81 GABRA1 (0.58) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7400032 0.80 GABRA1 (0.57) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7481780 0.79 GABRA1 (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL31226187 0.78 GABRA1 (0.45) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7208520 0.76 GABRA1 (0.56) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7209133 0.76 GABRA1 (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7005633 0.75 GABRA1 (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7487597 0.75 GABRA1 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7480454 0.75 GABRA1 (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024245156-A1 HETEROCYCLIC COMPOUND ACTING AS α5-GABAA RECEPTOR REGULATOR 武汉人福创新药物研发中心有限公司 2024-12-05 WO disclosed
CN-119019425-A Alpha 5-GABAAHeterocyclic compounds as receptor modulators 武汉人福创新药物研发中心有限公司 2024-11-26 CN disclosed