SCHEMBL31258474

SCHEMBL31258474

COc1cc2ncnc(Cl)c2cc1OC12CCCC(CC1)N2C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 5/20 0.43
EHMT2 Q96KQ7 2/20 0.40
EPHA2 P29317 7/20 0.39
EPHB4 P54760 5/20 0.39
KDR P35968 4/20 0.39
ERBB2 P04626 2/20 0.39
PIK3CD O00329 2/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CB P42338 2/20 0.38
PIK3CG P48736 2/20 0.38
MAPK7 Q13164 1/20 0.38
MAPK1 P28482 1/20 0.36
RAF1 P04049 1/20 0.36
BRAF P15056 1/20 0.36
NSD2 O96028 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31258476 0.85 PIK3CD (0.37) EPHA2EPHB4KDRERBB2PIK3CD
SCHEMBL30264691 0.79 EPHA2 (0.46) ENPP1EPHA2EPHB4KDRERBB2
SCHEMBL30639974 0.77 ERBB2 (0.49) ENPP1EPHA2EPHB4KDRERBB2
SCHEMBL31377604 0.77 ERBB2 (0.49) ENPP1EPHA2EPHB4KDRERBB2
SCHEMBL30639977 0.77 ERBB2 (0.49) ENPP1EPHA2EPHB4KDRERBB2
SCHEMBL665187 0.76 PIK3CD (0.54) EPHA2EPHB4KDRERBB2PIK3CD
SCHEMBL29465791 0.76 PIK3CD (0.54) EPHA2EPHB4KDRERBB2PIK3CD
SCHEMBL29465790 0.76 PIK3CD (0.54) EPHA2EPHB4KDRERBB2PIK3CD
SCHEMBL2453138 0.76 PIK3CD (0.54) EPHA2EPHB4KDRERBB2PIK3CD
SCHEMBL22598590 0.75 PIK3CD (0.51) ENPP1EHMT2EPHA2EPHB4ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118715216-A Nitrogen-containing heterocyclic compound, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2024-09-27 CN disclosed