SCHEMBL31276992

SCHEMBL31276992

N#Cc1cc(C=O)ccc1Oc1ccnc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.41
AAK1 Q2M2I8 1/20 0.41
SCN9A Q15858 8/20 0.40
SLC22A12 Q96S37 3/20 0.40
AR P10275 3/20 0.40
KDR P35968 2/20 0.39
ESRRA P11474 1/20 0.39
BRAF P15056 1/20 0.38
EPAS1 Q99814 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14663488 1.00 CYP3A4 (0.41) CYP3A4AAK1SCN9ASLC22A12AR
SCHEMBL875698 0.83 SCN9A (0.44) SCN9ASLC22A12AREPAS1
SCHEMBL14662019 0.83 KDR (0.46) KDRBRAF
SCHEMBL31276719 0.83 KDR (0.46) KDRBRAF
SCHEMBL15813965 0.83 SLC22A12 (0.40) SLC22A12ESRRA
SCHEMBL14662745 0.81 SLC22A12 (0.42) SLC22A12KDRESRRA
SCHEMBL17460293 0.81 TTR (0.41) CYP3A4AAK1SLC22A12ARESRRA
SCHEMBL15832066 0.81 AR (0.49) CYP3A4AAK1SLC22A12AR
SCHEMBL875764 0.81 SLC22A12 (0.39) SLC22A12ARESRRAEPAS1
SCHEMBL14662670 0.80 AR (0.61) ARESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119161343-A Bridged pyrimidinone compounds, preparation method thereof, pharmaceutical composition and application thereof 上海深势唯思科技有限责任公司 2024-12-20 CN disclosed
CN-119143780-A Lp-PLA2 inhibitor, preparation method thereof, pharmaceutical composition and application thereof 上海深势唯思科技有限责任公司 2024-12-17 CN disclosed
CN-119080800-A Tricyclic pyrimidinone compounds, preparation method thereof, pharmaceutical composition and application thereof 上海深势唯思科技有限责任公司 2024-12-06 CN disclosed