SCHEMBL31296544

SCHEMBL31296544

COC(=O)c1ccc(OC)cn1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.65
DYRK1A Q13627 1/20 0.53
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
KDM4E B2RXH2 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
P4HTM Q9NXG6 3/20 0.48
DRD3 P35462 1/20 0.46
MAPT P10636 3/20 0.44
POLB P06746 2/20 0.44
LCK P06239 1/20 0.44
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
ATM Q13315 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545257 1.00 MAPK1 (0.65) MAPK1DYRK1ACA1CA2KDM4E
SCHEMBL17007009 0.90 MAPK1 (0.57) MAPK1DYRK1ACA1CA2KDM4E
SCHEMBL13075575 0.85 MAPK1 (0.61) MAPK1DYRK1ACA1CA2KDM4E
SCHEMBL24969494 0.85 MAPK1 (0.61) MAPK1DYRK1ACA1CA2KDM4E
SCHEMBL15994646 0.85 MAPK1 (0.47) MAPK1DYRK1ACA1CA2KDM4E
SCHEMBL31620610 0.84 MAPK1 (0.59) MAPK1DYRK1AKDM4EL3MBTL1P4HTM
SCHEMBL10270980 0.84 MAPK1 (0.59) MAPK1DYRK1AKDM4EL3MBTL1P4HTM
SCHEMBL30827080 0.83 MAPK1 (0.54) MAPK1DYRK1AKDM4EL3MBTL1MAPT
SCHEMBL22529696 0.83 MAPK1 (0.54) MAPK1DYRK1AKDM4EL3MBTL1MAPT
SCHEMBL2187078 0.82 DRD3 (0.47) MAPK1CA1CA2KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119137107-A Macrocyclic inhibitors of ATP citrate lyase 艾斯柏伦治疗公司 2024-12-13 CN disclosed