SCHEMBL313272

SCHEMBL313272

CCN(O)C(CS)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.36
SLC7A11 Q9UPY5 1/20 0.36
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
ALOX15 P16050 1/20 0.34
NFKB1 P19838 1/20 0.34
PTGS2 P35354 1/20 0.34
THPO P40225 1/20 0.34
RECQL P46063 1/20 0.34
BLM P54132 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ENPEP Q07075 4/20 0.33
ACE P12821 1/20 0.31
FOLH1 Q04609 1/20 0.31
CHRM1 P11229 1/20 0.31
AKR1A1 P14550 1/20 0.31
CHRM3 P20309 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL898887 1.00 PTGS1 (0.36) PTGS1SLC7A11KDM4EMAPTTHRB
SCHEMBL313183 0.83 FOLH1 (0.36) ENPEPFOLH1CHRM1AKR1A1CHRM3
SCHEMBL5961754 0.83 FOLH1 (0.36) ENPEPFOLH1CHRM1AKR1A1CHRM3
SCHEMBL3728136 0.81 CHRM1 (0.33) CHRM1AKR1A1CHRM3HTR2AHTR2C
SCHEMBL19737260 0.79 PTGS1 (0.37) PTGS1SLC7A11KDM4EMAPTTHRB
SCHEMBL20512314 0.79 PTGS1 (0.37) PTGS1SLC7A11KDM4EMAPTTHRB
SCHEMBL17772932 0.77 PTGS1 (0.36) PTGS1SLC7A11KDM4EMAPTTHRB
SCHEMBL7150005 0.77 PTGS1 (0.36) PTGS1SLC7A11KDM4EMAPTTHRB
SCHEMBL11584178 0.77 PTGS1 (0.36) PTGS1SLC7A11KDM4EMAPTTHRB
SCHEMBL8407151 0.77 TDP1 (0.39) MAPTSMN1; SMN2FOLH1CHRM1AKR1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2182 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11203622-B2 MASP isoforms as inhibitors of complement activation OMEROS CORPORATION (US) 2021-12-21 US claimed
EP-2688578-B1 MIA (MELANOMA INHIBITORY ACTIVITY) INHIBITORS FOR PREVENTING AND CURING VITILIGO BORDIGNON MATTEO (IT) 2019-03-27 EP claimed
EP-2688578-A2 MIA (MELANOMA INHIBITORY ACTIVITY) INHIBITORS FOR DETECTING, PREVENTING AND CURING VITILIGO Bordignon, Matteo (IT) 2014-01-29 EP claimed
US-20140004130-A1 MIA (Melanoma Inhibitory Activity) Inhibitors for Detecting, Preventing and Curing Vitiligo BORDIGNON MATTEO (IT) 2014-01-02 US claimed
WO-2012127352-A2 MIA (MELANOMA INHIBITORY ACTIVITY) INHIBITORS FOR DETECTING, PREVENTING AND CURING VITILIGO BORDIGNON MATTEO (IT) 2012-09-27 WO claimed
US-20120208774-A1 METHOD FOR INHIBITING \"MELANOMA INHIBITORY ACTIVITY\" MIA ANTISENSE PHARMA GMBH (DE) 2012-08-16 US claimed
US-8148493-B2 Method for inhibiting “melanoma inhibitory activity” MIA ANTISENSE PHARMA GMBH (DE) 2012-04-03 US claimed
US-20100273705-A1 Method for inhibiting \"Melanoma Inhibitory Activity\" MIA ANTISENSE PHARMA GMBH. 2010-10-28 US claimed
US-20060128607-A1 Method for inhibiting \"melanoma inhibitory activity\" mia ANTISENSE PHARMA GMBH (DE) 2006-06-15 US claimed
US-20260146104-A1 ANTIBODIES, ACTIVATABLE ANTIBODIES, BISPECIFIC ANTIBODIES, AND BISPECIFIC ACTIVATABLE ANTIBODIES AND METHODS OF USE THEREOF CYTOMX THERAPEUTICS, INC. (US) 2026-05-28 US disclosed
US-20260115317-A1 GENE THERAPY IMPERIAL COLLEGE INNOVATIONS LTD (GB) 2026-04-30 US disclosed
US-20260103454-A1 MODULATORS OF HEMOGLOBIN GLOBAL BLOOD THERAPEUTICS INC (US) 2026-04-16 US disclosed
EP-3890772-B1 BOTULINUM TOXIN FOR USE IN THE TREATMENT OF SYMPTOMS OF TRAUMATIC BRAIN INJURY IPSEN BIOPHARM LTD (GB) 2026-04-01 EP disclosed
US-12589139-B2 Clostridial neurotoxins comprising an exogenous activation loop IPSEN BIOPHARM LIMITED (GB) 2026-03-31 US disclosed
WO-1998029419-A1 CYANOPHOSPHORUS COMPOUNDS AND THEIR PREPARATION MONSANTO COMPANY (US) 1998-07-09 WO disclosed
WO-1998029422-A1 CYANOPHOSPHONATE DERIVATIVES MONSANTO COMPANY (US) 1998-07-09 WO disclosed
WO-1998027210-A1 COMPOSITIONS AND METHODS FOR STIMULATING PANCREATIC ISLET CELL REGENERATION ZYMOGENETICS, INC. (US) 1998-06-25 WO disclosed
WO-1998016635-A1 INSULIN HOMOLOGS ZYMOGENETICS, INC. (US) 1998-04-23 WO disclosed
WO-1998016644-A1 FIBROBLAST GROWTH FACTOR HOMOLOGS ZYMOGENETICS, INC. (US) 1998-04-23 WO disclosed
WO-1998005782-A1 TESTIS-SPECIFIC INSULIN HOMOLOG POLYPEPTIDES ZYMOGENETICS, INC. (US) 1998-02-12 WO disclosed