SCHEMBL3133467

SCHEMBL3133467

CC(C)(NC(=O)OC1CC(c2cc(NC(=O)C3CCOCC3)n[nH]2)C1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 20/20 0.49
CCNE1 P24864 19/20 0.49
GSK3B P49841 13/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3133459 1.00 CDK2 (0.49) CDK2CCNE1GSK3B
SCHEMBL3130801 0.79 CDK2 (0.49) CDK2CCNE1GSK3B
SCHEMBL3125245 0.79 CDK2 (0.53) CDK2CCNE1GSK3B
SCHEMBL3125243 0.79 CDK2 (0.53) CDK2CCNE1GSK3B
SCHEMBL3130806 0.79 CDK2 (0.49) CDK2CCNE1GSK3B
SCHEMBL3564951 0.79 CDK2 (0.47) CDK2CCNE1GSK3B
SCHEMBL25938137 0.75 CDK2 (0.67) CDK2CCNE1GSK3B
SCHEMBL25941301 0.75 CDK2 (0.67) CDK2CCNE1GSK3B
SCHEMBL3134085 0.75 CDK2 (0.54) CDK2CCNE1GSK3B
SCHEMBL3134092 0.75 CDK2 (0.54) CDK2CCNE1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689721-B1 AMINOPYRAZOLE DERIVATIVES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2010-07-14 EP claimed
US-7671072-B2 Aminopyrazole derivatives as GSK-3 inhibitors PFIZER INC. (US) 2010-03-02 US claimed
EP-1689721-B1 AMINOPYRAZOLE DERIVATIVES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2010-07-14 EP disclosed