SCHEMBL31363591

SCHEMBL31363591

NC(=O)c1cccc2c1ncn2CC(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 4/20 0.51
CYP1A2 P05177 1/20 0.48
PARP1 P09874 9/20 0.42
AR P10275 3/20 0.40
PARP2 Q9UGN5 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
PARP3 Q9Y6F1 1/20 0.38
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
AURKB Q96GD4 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28634932 0.83 CYP17A1 (0.48) CYP17A1CYP1A2AREGLN1
SCHEMBL1290332 0.78 PARP1 (0.47) PARP1L3MBTL1AURKARPS6KB1AURKB
SCHEMBL30119632 0.78 CYP17A1 (0.60) CYP17A1CYP1A2ARL3MBTL1
SCHEMBL29829828 0.76 HTT (0.54) PARP1PARP2PARP3AURKARPS6KB1
SCHEMBL21555726 0.75 CYP17A1 (0.54) CYP17A1CYP1A2AR
SCHEMBL28625938 0.75 CYP17A1 (0.51) CYP17A1CYP1A2AR
SCHEMBL30098925 0.74 IDO1 (0.44) L3MBTL1
SCHEMBL16497015 0.74 PARP1 (0.49) PARP1PARP2L3MBTL1PARP3AURKA
SCHEMBL29830638 0.74 ADRA1D (0.48) PARP1PARP2PARP3AURKARPS6KB1
SCHEMBL27249587 0.73 PARP1 (0.47) PARP1L3MBTL1AURKARPS6KB1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025059074-A1 BICYCLIC COMPOUNDS FOR RESTORING MUTANT P53 FUNCTION PMV PHARMACEUTICALS, INC. (US) 2025-03-20 WO disclosed