SCHEMBL31367342

SCHEMBL31367342

COC(=O)c1cc2c(cc1F)CC=C2c1ccccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CFTR P13569 5/20 0.39
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PDK2 Q15119 3/20 0.36
SDHB P21912 1/20 0.36
RBP4 P02753 1/20 0.36
BDKRB1 P46663 1/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
LDHA P00338 1/20 0.35
NOTUM Q6P988 1/20 0.34
PTK2 Q05397 1/20 0.34
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17276115 1.00 CFTR (0.39) CFTRSLC6A4SLC6A3AKR1C3AKR1C2
SCHEMBL17276219 0.81 PDK2 (0.50) SMN1; SMN2PDK2RBP4NOTUM
SCHEMBL31367303 0.77 PDK2 (0.46) CFTRSLC6A4SLC6A3AKR1C3AKR1C2
SCHEMBL17276328 0.77 PDK2 (0.46) CFTRSLC6A4SLC6A3AKR1C3AKR1C2
SCHEMBL17276275 0.76 PDK2 (0.45) CFTRSLC6A4SLC6A3AKR1C3AKR1C2
SCHEMBL12389765 0.73 PDK2 (0.48) ALDH1A1HPGDSMN1; SMN2PDK2RBP4
SCHEMBL28133503 0.71 PDK2 (0.36) ALDH1A1HPGDPDK2RBP4LMNA
SCHEMBL17276098 0.70 NR4A2 (0.44) CFTRSLC6A4SLC6A3AKR1C3AKR1C2
SCHEMBL28841543 0.70 APP (0.41) AKR1C3AKR1C2ALDH1A1HPGD
SCHEMBL28134284 0.70 HSD11B1 (0.40) ALDH1A1HPGDNOTUMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3145915-B1 ANTIDIABETIC TRICYCLIC COMPOUNDS MERCK SHARP & DOHME LLC (US) 2025-03-19 EP disclosed