SCHEMBL3141014

SCHEMBL3141014

C=CN1C=CC(=O)C1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10703046 0.64 HDAC3 (0.35)
SCHEMBL295379 0.62
SCHEMBL2802598 0.62
SCHEMBL11003248 0.62
SCHEMBL9887684 0.60
SCHEMBL9187467 0.60
SCHEMBL28975614 0.59
SCHEMBL6365325 0.57
Hydrochloric Acid SCHEMBL28977690 0.56
SCHEMBL895297 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11752100-B2 Intranasal delivery of olanzapine by precision olfactory device IMPEL PHARMACEUTICALS INC. (US) 2023-09-12 US claimed
US-20220183965-A1 INTRANASAL DELIVERY OF OLANZAPINE BY PRECISION OLFACTORY DEVICE ALTER DOMUS (US) LLC 2022-06-16 US claimed
US-11278492-B2 Intranasal delivery of olanzapine by precision olfactory device IMPEL NEUROPHARMA, INC. (US) 2022-03-22 US claimed
EP-1379367-A4 WATER SOLUBLE TOOLING MATERIALS FOR COMPOSITE STRUCTURES ADVANCED CERAMICS RES INC (US) 2004-06-23 EP claimed
EP-1379367-A1 WATER SOLUBLE TOOLING MATERIALS FOR COMPOSITE STRUCTURES Advanced Ceramics Research, Inc. (US) 2004-01-14 EP claimed
US-20020173575-A1 Water soluble tooling materials for composite structures ADVANCED CERAMICS RESEARCH LLC 2002-11-21 US claimed
WO-2002072328-A1 WATER SOLUBLE TOOLING MATERIALS FOR COMPOSITE STRUCTURES ADVANCED CERAMICS RESEARCH, INC. (US) 2002-09-19 WO claimed
US-20240252489-A1 REPEATED ADMINISTRATION OF DIHYDROERGOTAMINE FOR TREATMENT OF FREQUENT MIGRAINE HEADACHES ALTER DOMUS (US) LLC 2024-08-01 US disclosed
US-20230364010-A1 INTRANASAL DELIVERY OF OLANZAPINE BY PRECISION OLFACTORY DEVICE WOODWARD SPECIALTY LLC (PR) 2023-11-16 US disclosed
US-11752100-B2 Intranasal delivery of olanzapine by precision olfactory device IMPEL PHARMACEUTICALS INC. (US) 2023-09-12 US disclosed
EP-4090331-A1 REPEATED ADMINISTRATION OF DIHYDROERGOTAMINE FOR TREATMENT OF FREQUENT MIGRAINE HEADACHES Impel Pharmaceuticals Inc. (US) 2022-11-23 EP disclosed
CN-115279371-A Repeated administration of dihydroergotamine for the treatment of frequent migraine 英倍尔制药公司 2022-11-01 CN disclosed
US-20220183965-A1 INTRANASAL DELIVERY OF OLANZAPINE BY PRECISION OLFACTORY DEVICE ALTER DOMUS (US) LLC 2022-06-16 US disclosed
WO-2002072328-A1 WATER SOLUBLE TOOLING MATERIALS FOR COMPOSITE STRUCTURES ADVANCED CERAMICS RESEARCH, INC. (US) 2002-09-19 WO disclosed
US-6086854-A Antiplaque oral composition ARNOLD MICHAEL J (US) 2000-07-11 US disclosed
EP-0921783-B1 ANTIPLAQUE ORAL COMPOSITION ARNOLD MICHAEL J (US) 2000-03-22 EP disclosed
US-5804165-A TABLET OR CAPSULE CONTAINING EFFERVESCENT POWDER COMPRISING NONAQUEOUS, WATER SOLUBLE CARBONATE AND/OR BICARBONATE SALT, SILICA, AND XYLITOL; GOOD TASTE, NONTOXIC, EFFICIENCY 90 SECONDS TO WOW, LLC 1998-09-08 US disclosed
CN-1163780-A Osteogenesis stimulin injection and its preparing process WHOLE ARMY INST OF TRAUMATOLOG (CN) 1997-11-05 CN disclosed
CN-1124788-A Pickling paste for stainless steel SUN YONGCHUN (CN) 1996-06-19 CN disclosed
US-5326683-A Black and white reverse image, hydrazine nucleating agent, redox compound FUJI PHOTO FILM CO., LTD. (JP) 1994-07-05 US disclosed