SCHEMBL31415917

SCHEMBL31415917

COC1(OC)CC(NC(=O)OCc2ccccc2)C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
GAA P10253 1/20 0.59
TSHR P16473 2/20 0.56
EPHX1 P07099 1/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
ACHE P22303 2/20 0.52
CPB1 P15086 1/20 0.51
CTSL P07711 1/20 0.51
CTSB P07858 1/20 0.51
CTSK P43235 1/20 0.51
ROCK2 O75116 1/20 0.48
ENPP2 Q13822 1/20 0.48
ATXN2 Q99700 1/20 0.48
CYP3A4 P08684 1/20 0.48
CASP1 P29466 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TLR4 O00206 1/20 0.47
KDM1A O60341 1/20 0.47
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21945637 0.88 ALDH1A1 (0.58) ALDH1A1GAATSHREPHX1CA1
SCHEMBL25190914 0.87 KMT2A (0.50) ALDH1A1GAATSHREPHX1CA1
SCHEMBL6758979 0.86 ALDH1A1 (0.62) ALDH1A1GAATSHREPHX1CA1
SCHEMBL21945751 0.84 ALDH1A1 (0.60) ALDH1A1GAATSHREPHX1CA1
SCHEMBL21945750 0.84 ALDH1A1 (0.60) ALDH1A1GAATSHREPHX1CA1
SCHEMBL21946019 0.84 ALDH1A1 (0.60) ALDH1A1GAATSHREPHX1CA1
SCHEMBL361720 0.83 ALDH1A1 (0.62) ALDH1A1GAATSHREPHX1CA1
SCHEMBL31641122 0.82 ALDH1A1 (0.58) ALDH1A1GAATSHREPHX1CA1
SCHEMBL28567212 0.82 EZH2 (0.60) ALDH1A1GAATSHREPHX1ENPP2
SCHEMBL10196993 0.82 ALDH1A1 (0.60) ALDH1A1GAATSHREPHX1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4735444-A1 BENZYL (3-(METHYL(7H-PYRROLO[2,3-D]PYRIMIDIN-4YL)AMINO)CYCLOBUTYL) CARBAMATE OR A SALT THEREOF, METHOD FOR THE PREPARATION THEREOF, AND USE THEREOF IN THE SYNTHESIS OF ABROCITINIB Moehs Ibérica, S.L. (ES) 2026-05-06 EP disclosed
WO-2025003177-A1 BENZYL (3-(METHYL(7H-PYRROLO[2,3-D]PYRIMIDIN-4YL)AMINO)CYCLOBUTYL) CARBAMATE OR A SALT THEREOF, METHOD FOR THE PREPARATION THEREOF, AND USE THEREOF IN THE SYNTHESIS OF ABROCITINIB MOEHS IBERICA, S.L. (ES) 2025-01-02 WO disclosed