SCHEMBL3141865

SCHEMBL3141865

COc1ccc2ccc(Br)c(CC#N)c2n1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.45
DYRK1A Q13627 1/20 0.45
MTNR1A P48039 15/20 0.34
MTNR1B P49286 15/20 0.34
HTR2C P28335 3/20 0.32
PTGS2 P35354 1/20 0.31
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1712036 0.82 CLK1 (0.45) CLK1DYRK1AMTNR1AMTNR1BHTR2C
SCHEMBL1712516 0.81 MTNR1A (0.37) MTNR1AMTNR1BHTR2CPTGS2NQO2
SCHEMBL1712254 0.81 MTNR1A (0.37) MTNR1AMTNR1BHTR2CPTGS2NQO2
SCHEMBL1712179 0.80 MTNR1A (0.39) MTNR1AMTNR1BHTR2CPTGS2
SCHEMBL28792431 0.78 MTNR1A (0.38) MTNR1AMTNR1BHTR2CPTGS2NQO2
SCHEMBL3149015 0.75 MTNR1A (0.41) MTNR1AMTNR1BHTR2CPTGS2
SCHEMBL3142042 0.72 NQO2 (0.38) MTNR1AMTNR1BHTR2CNQO2
SCHEMBL31575293 0.71 CLK1 (0.39) CLK1DYRK1A
SCHEMBL23208944 0.70 MTNR1A (0.35) MTNR1AMTNR1BHTR2CNQO2
SCHEMBL29970846 0.70 MTNR1A (0.35) MTNR1AMTNR1BHTR2CNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954697-B1 PERI CONDENSED TRICYCLIC COMPOUNDS USEFUL AS ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2010-02-24 EP disclosed