SCHEMBL3143603

SCHEMBL3143603

[CH2]c1cnn(-c2cccc(F)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.50
GRM4 Q14833 2/20 0.49
KEAP1 Q14145 1/20 0.47
NOTUM Q6P988 1/20 0.45
MTOR P42345 1/20 0.44
EPHX2 P34913 1/20 0.42
RXRA P19793 6/20 0.42
GRIN1 Q05586 6/20 0.42
GRIN2B Q13224 6/20 0.42
FAAH O00519 1/20 0.40
MGLL Q99685 1/20 0.40
ADORA3 P0DMS8 2/20 0.39
RAB9A P51151 1/20 0.39
ADORA2A P29274 1/20 0.39
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3143610 0.79 NPC1 (0.50) NPC1GRM4KEAP1NOTUMMTOR
SCHEMBL27638750 0.79 NPC1 (0.50) NPC1GRM4KEAP1NOTUMMTOR
SCHEMBL1304053 0.77 GAA (0.59) NPC1GRM4MTORRAB9AGAA
SCHEMBL15181516 0.76 MTOR (0.56) NPC1GRM4KEAP1NOTUMMTOR
SCHEMBL18878403 0.76 NPC1 (0.47) NPC1GRM4KEAP1NOTUMMTOR
SCHEMBL19249155 0.76 NPC1 (0.50) NPC1GRM4KEAP1NOTUMMTOR
SCHEMBL2411161 0.76 NPC1 (0.47) NPC1GRM4KEAP1NOTUMMTOR
SCHEMBL26054257 0.76 NPC1 (0.47) NPC1GRM4KEAP1NOTUMMTOR
SCHEMBL4796959 0.74 ALKBH2 (0.69) NPC1KEAP1RAB9A
SCHEMBL20729400 0.72 NPC1 (0.44) NPC1GRM4KEAP1NOTUMMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233493-A1 Macrolides Pfizer Products Inc. (US) 2010-09-29 EP disclosed
EP-1836211-B1 MACROLIDES PFIZER PROD INC (US) 2010-03-03 EP disclosed