SCHEMBL3145014

SCHEMBL3145014

CCCCCc1ccc(NC(=S)NC(=O)c2ccc3oc(C(=O)O)cc3c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 6/20 0.54
SIRT1 Q96EB6 6/20 0.54
MAPT P10636 3/20 0.49
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2864487 0.89 SIRT2 (0.51) SIRT2SIRT1MAPTNPC1RAB9A
SCHEMBL13971438 0.84 MAPT (0.56) SIRT2SIRT1MAPTNPC1RAB9A
SCHEMBL5839894 0.83 MAPT (0.55) SIRT2SIRT1MAPTNPC1RAB9A
SCHEMBL13956740 0.82 MAPT (0.73) MAPTNPC1RAB9AALDH1A1MEN1
SCHEMBL4364678 0.81 MAPT (0.52) SIRT2SIRT1MAPTNPC1RAB9A
SCHEMBL4363295 0.80 MAPT (0.52) SIRT2SIRT1MAPTNPC1RAB9A
SCHEMBL13971233 0.79 MAPT (0.74) MAPTNPC1RAB9AALDH1A1MEN1
SCHEMBL13175624 0.78 ALDH1A1 (0.54) SIRT2SIRT1MAPTNPC1RAB9A
Hydrochloric Acid SCHEMBL3718452 0.78 SIRT2 (0.67) SIRT2SIRT1MAPTTDP1ALDH1A1
Hydrochloric Acid SCHEMBL3718449 0.78 SIRT2 (0.67) SIRT2SIRT1MAPTTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747196-B1 SUBSTITUTED ARYL ACYLTHIOUREAS AND RELATED COMPOUNDS; INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS INC (US) 2010-02-10 EP claimed