SCHEMBL3145250

SCHEMBL3145250

NCC1(COc2cnc(Cl)c(-c3cccc(-c4nn[nH]n4)c3)c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
GP6 Q9HCN6 2/20 0.40
SLC22A12 Q96S37 2/20 0.39
CREBBP Q92793 1/20 0.39
MRGPRX4 Q96LA9 2/20 0.39
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37
HPGDS O60760 1/20 0.37
CYSLTR2 Q9NS75 1/20 0.36
CYSLTR1 Q9Y271 1/20 0.36
ALDH1A1 P00352 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
XDH P47989 1/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3774366 0.99 IDO1 (0.41) IDO1GP6SLC22A12CREBBPMRGPRX4
SCHEMBL3150837 0.91 MAP4K4 (0.43) MRGPRX4HPGDSALDH1A1XDHMAP4K4
Hydrochloric Acid SCHEMBL3154957 0.90 MAP4K4 (0.43) MRGPRX4HPGDSALDH1A1XDHMAP4K4
SCHEMBL3151049 0.85 EGLN1 (0.43) IDO1GP6SLC22A12CREBBPEGLN1
Hydrochloric Acid SCHEMBL3774374 0.83 IDO1 (0.40) IDO1GP6SLC22A12CREBBPMRGPRX4
SCHEMBL3155932 0.82 DHFR (0.39)
SCHEMBL3777217 0.81 CREBBP (0.40) IDO1GP6SLC22A12CREBBPEGLN1
SCHEMBL3154920 0.81 MAP4K4 (0.35) MAP4K4
Hydrochloric Acid SCHEMBL3767963 0.81 DHFR (0.38)
SCHEMBL3155946 0.81 FFAR4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed