SCHEMBL3149677

SCHEMBL3149677

CC(C)c1nnn(-c2c(F)cccc2Cl)c1COc1ccc(-c2ccc(C(=O)O)cc2)c(Cl)c1

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 19/20 0.63
VDR P11473 2/20 0.41
SRD5A2 P31213 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3165576 0.94 NR1H4 (0.70) NR1H4VDRSRD5A2
SCHEMBL3150919 0.94 NR1H4 (0.61) NR1H4VDR
SCHEMBL3155021 0.92 NR1H4 (0.67) NR1H4VDR
SCHEMBL498129 0.87 NR1H4 (0.68) NR1H4VDR
SCHEMBL498287 0.87 NR1H4 (0.67) NR1H4VDRSRD5A2
SCHEMBL3169067 0.86 NR1H4 (0.65) NR1H4VDRSRD5A2
SCHEMBL3168275 0.84 NR1H4 (0.64) NR1H4VDRSRD5A2
SCHEMBL3162062 0.82 NR1H4 (0.52) NR1H4VDRSRD5A2
SCHEMBL498488 0.81 NR1H4 (0.54) NR1H4
SCHEMBL3165823 0.81 NR1H4 (0.51) NR1H4VDRSRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029558-B1 COMPOUNDS AND METHODS FOR MODULATING FXR LILLY CO ELI (US) 2010-03-10 EP disclosed