SCHEMBL498488

SCHEMBL498488

CC(=O)c1ccc(OCc2c(C(C)C)nnn2-c2c(F)cccc2Cl)cc1C

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.54
MAOB P27338 6/20 0.41
MAOA P21397 3/20 0.39
KMT2A Q03164 1/20 0.36
RAB9A P51151 1/20 0.35
DHODH Q02127 2/20 0.35
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497577 0.94 NR1H4 (0.60) NR1H4MAOBMAOAKMT2AALDH1A1
SCHEMBL498015 0.86 NR1H4 (0.51) NR1H4KMT2ARAB9ADHODHL3MBTL1
SCHEMBL3150919 0.85 NR1H4 (0.61) NR1H4
SCHEMBL3150227 0.81 NR1H4 (0.59) NR1H4RAB9A
SCHEMBL3149677 0.81 NR1H4 (0.63) NR1H4
SCHEMBL498233 0.81 NR1H4 (0.62) NR1H4MAOBMAOAALDH1A1MAPT
SCHEMBL3164115 0.81 NR1H4 (0.79) NR1H4KMT2A
SCHEMBL3164111 0.81 NR1H4 (0.79) NR1H4KMT2A
SCHEMBL498760 0.80 NR1H4 (0.58) NR1H4
SCHEMBL498759 0.79 NR1H4 (0.57) NR1H4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106077-B2 Compounds and methods for modulating FXR ELI LILLY AND COMPANY (US) 2012-01-31 US disclosed
EP-2029558-B1 COMPOUNDS AND METHODS FOR MODULATING FXR LILLY CO ELI (US) 2010-03-10 EP disclosed