SCHEMBL3149728

SCHEMBL3149728

Cc1cc(OCc2c(C(C)C)nnn2-c2c(Cl)cccc2Cl)ccc1C(C)Oc1cccc(CCC(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.52
FFAR1 O14842 16/20 0.39
FFAR4 Q5NUL3 3/20 0.37
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3159265 0.92 NR1H4 (0.54) NR1H4PPARD
SCHEMBL3150227 0.82 NR1H4 (0.59) NR1H4PPARG
SCHEMBL498139 0.81 NR1H4 (0.57) NR1H4
SCHEMBL497577 0.77 NR1H4 (0.60) NR1H4
SCHEMBL497776 0.76 NR1H4 (0.63) NR1H4
SCHEMBL498015 0.75 NR1H4 (0.51) NR1H4
SCHEMBL497662 0.75 NR1H4 (0.56) NR1H4
SCHEMBL498491 0.75 NR1H4 (0.64) NR1H4
SCHEMBL498129 0.75 NR1H4 (0.68) NR1H4
SCHEMBL498302 0.74 NR1H4 (0.60) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029558-B1 COMPOUNDS AND METHODS FOR MODULATING FXR LILLY CO ELI (US) 2010-03-10 EP disclosed