SCHEMBL3159265

SCHEMBL3159265

Cc1cc(OCc2c(C(C)C)nnn2-c2c(Cl)cccc2Cl)ccc1C(C)Oc1cccc(CC(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 13/20 0.54
PPARD Q03181 6/20 0.37
MRGPRX4 Q96LA9 1/20 0.36
KMT2A Q03164 1/20 0.36
CCNK O75909 1/20 0.33
CCND3 P30281 1/20 0.33
GSK3B P49841 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
CCNH P51946 1/20 0.33
CDK6 Q00534 1/20 0.33
CDK12 Q9NYV4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3149728 0.92 NR1H4 (0.52) NR1H4PPARD
SCHEMBL3150227 0.84 NR1H4 (0.59) NR1H4MRGPRX4
SCHEMBL498139 0.82 NR1H4 (0.57) NR1H4MRGPRX4KMT2ACCNKCCND3
SCHEMBL3165066 0.81 NR1H4 (0.51) NR1H4PPARDMRGPRX4KMT2A
SCHEMBL3165073 0.81 NR1H4 (0.51) NR1H4PPARDMRGPRX4KMT2A
SCHEMBL497577 0.79 NR1H4 (0.60) NR1H4MRGPRX4KMT2ACCNKCCND3
SCHEMBL3150710 0.79 NR1H4 (0.53) NR1H4PPARDMRGPRX4KMT2ACCNK
SCHEMBL3150714 0.79 NR1H4 (0.51) NR1H4PPARDKMT2ACCNKCCND3
SCHEMBL3157598 0.78 NR1H4 (0.52) NR1H4PPARDMRGPRX4
SCHEMBL3157584 0.77 NR1H4 (0.53) NR1H4PPARDMRGPRX4CCNKCCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029558-B1 COMPOUNDS AND METHODS FOR MODULATING FXR LILLY CO ELI (US) 2010-03-10 EP disclosed