SCHEMBL315424

SCHEMBL315424

Cc1ccccc1CC1(N(C)C)CCC(NC(=O)c2c(-c3c(Cl)cccc3Cl)noc2C)CC1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 5/20 0.61
KMT2A Q03164 2/20 0.53
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
PTGS2 P35354 2/20 0.48
TSHR P16473 1/20 0.47
GLA P06280 1/20 0.46
PKM P14618 1/20 0.46
POLB P06746 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316040 0.95 GHSR (0.55) GHSRKMT2AALDH1A1MAPTGLA
SCHEMBL316283 0.95 GHSR (0.62) GHSRKMT2AALDH1A1KDM4EGAA
SCHEMBL316058 0.92 KMT2A (0.65) GHSRKMT2AALDH1A1MAPTTDP1
SCHEMBL315545 0.91 GHSR (0.59) GHSRKMT2AALDH1A1KDM4EGAA
SCHEMBL316102 0.90 GHSR (0.56) GHSRKMT2AALDH1A1MAPTPOLB
SCHEMBL314979 0.89 GHSR (0.62) GHSRKMT2AALDH1A1KDM4EGAA
SCHEMBL315422 0.87 GHSR (0.61) GHSRKMT2AALDH1A1KDM4EGAA
SCHEMBL316492 0.87 GHSR (0.61) GHSRKMT2AALDH1A1KDM4EGAA
SCHEMBL315886 0.85 GHSR (0.60) GHSRKMT2AALDH1A1KDM4EGAA
SCHEMBL316299 0.84 KMT2A (0.57) GHSRKMT2AALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed