SCHEMBL3166124

SCHEMBL3166124

O=C(O)C1(c2ccccc2I)CCC(OCC2CC2)(c2ccnc(-c3ccccc3)c2)CC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
F11 P03951 1/20 0.33
PDE4D Q08499 4/20 0.33
KMO O15229 2/20 0.32
NR1H4 Q96RI1 1/20 0.32
VCP P55072 1/20 0.32
KAT6A Q92794 1/20 0.31
ADAM17 P78536 1/20 0.31
WNT3A P56704 1/20 0.31
CNR1 P21554 1/20 0.30
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
KDM5A P29375 1/20 0.30
KDM2B Q8NHM5 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3013594 0.88 ACACB (0.39) ACACBACACAF11PDE4DKMO
SCHEMBL3013591 0.88 ACACB (0.39) ACACBACACAF11PDE4DKMO
SCHEMBL3013597 0.88 ACACB (0.39) ACACBACACAF11PDE4DKMO
SCHEMBL3019314 0.73 NR1H4 (0.39) F11NR1H4CNR1
SCHEMBL3019312 0.73 NR1H4 (0.39) F11NR1H4CNR1
SCHEMBL3019311 0.73 NR1H4 (0.39) F11NR1H4CNR1
SCHEMBL3008631 0.69 AKR1C1 (0.41) KDM2B
SCHEMBL3019258 0.68 ELOVL1 (0.43)
SCHEMBL3018150 0.68 ERCC5 (0.38) NR1H4
SCHEMBL10528592 0.68 AKR1C1 (0.52) KDM2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164825-A1 DI(HETERO)ARYLCYCLOHEXANE DERIVATIVES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Sanofi-Aventis (FR) 2010-03-24 EP disclosed
WO-2008148468-A1 DI(HETERO)ARYLCYCLOHEXANE DERIVATIVES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM SANOFI-AVENTIS (FR) 2008-12-11 WO disclosed