SCHEMBL31676996

SCHEMBL31676996

O=c1cc(-c2cn[nH]c2)[nH]c2ncnn12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.34
FYN P06241 3/20 0.33
TDP1 Q9NUW8 1/20 0.33
ACVR1 Q04771 1/20 0.33
ALDH1A1 P00352 1/20 0.32
SIRT5 Q9NXA8 1/20 0.32
XDH P47989 1/20 0.32
AURKA O14965 6/20 0.32
CCNA2 P20248 6/20 0.32
CDK2 P24941 6/20 0.32
TTK P33981 6/20 0.32
KDM5B Q9UGL1 1/20 0.32
MAPKAPK5 Q8IW41 1/20 0.31
FGFR3 P22607 1/20 0.31
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
AURKB Q96GD4 2/20 0.31
CHEK1 O14757 2/20 0.31
CHEK2 O96017 2/20 0.31
ABL1 P00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31677033 0.81 TSHR (0.36) TSHRTDP1ALDH1A1SIRT5XDH
SCHEMBL20074201 0.77 CDC7 (0.40) TDP1ACVR1ALDH1A1CDK2MAPKAPK5
SCHEMBL20074294 0.76 KDM5B (0.40) TSHRACVR1AURKACCNA2CDK2
SCHEMBL20074198 0.76 KDM5B (0.44) TSHRAURKAKDM5BFGFR3AURKB
SCHEMBL20074296 0.75 CHEK1 (0.42) TSHRACVR1ALDH1A1AURKAKDM5B
SCHEMBL31677015 0.75 SMN1; SMN2 (0.45) ALDH1A1
SCHEMBL31676986 0.71 CDK8 (0.45) FYNACVR1CDK2KDM5BAURKB
SCHEMBL31677026 0.71 KDM5B (0.40) TSHRKDM5BFGFR3AURKB
SCHEMBL31677002 0.70 POLB (0.34) TSHRTDP1CCNA2CDK2TTK
SCHEMBL20074119 0.69 KDM5B (0.46) TSHRALDH1A1SIRT5KDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3525785-B1 KDM5 INHIBITORS MERCK SHARP & DOHME LLC (US) 2025-08-27 EP claimed